Structure–Activity Relationships of (+)-Naltrexone-Inspired Toll-like Receptor 4 (TLR4) Antagonists | Journal of Medicinal Chemistry
Design of Selective Benzoxazepin PI3Kδ Inhibitors Through Control of Dihedral Angles | ACS Medicinal Chemistry Letters
In Search of the Optimal Macrocyclization Site for Neurotensin | ACS Medicinal Chemistry Letters
Discovery of APD371: Identification of a Highly Potent and Selective CB2 Agonist for the Treatment of Chronic Pain | ACS Medicinal Chemistry Letters
Structure-Based Design of Inhibitors Selective for Human Proteasome β2c or β2i Subunits | Journal of Medicinal Chemistry
Structure and Mechanism-Guided Design of Dual Serine/Metallo-Carbapenemase Inhibitors | Journal of Medicinal Chemistry
Synthesis and Cell-Based Activity of a Potent and Selective Protein Tyrosine Phosphatase 1B Inhibitor Prodrug | Journal of Medicinal Chemistry
Rational Alteration of Pharmacokinetics of Chiral Fluorinated and Deuterated Derivatives of Emixustat for Retinal Therapy | Journal of Medicinal Chemistry
Forging Odd-Membered Rings: Palladium-Catalyzed Asymmetric Cycloadditions of Trimethylenemethane | Accounts of Chemical Research
Discovery of 5-Nitro-6-thiocyanatopyrimidines as Inhibitors of Cryptococcus neoformans and Cryptococcus gattii | ACS Medicinal Chemistry Letters
Scaffold-Hopping Strategy on a Series of Proteasome Inhibitors Led to a Preclinical Candidate for the Treatment of Visceral Leishmaniasis | Journal of Medicinal Chemistry
Stabilization of Nanoparticles Produced by Hydrogenation of Palladium–N-Heterocyclic Carbene Complexes on the Surface of Graphene and Implications in Catalysis | ACS Omega
ACS Medicinal Chemistry Letters | Vol 11, No 11
Design, Synthesis, and Structure–Activity Relationship Optimization of Pyrazolopyrimidine Amide Inhibitors of Phosphoinositide 3-Kinase γ (PI3Kγ) | Journal of Medicinal Chemistry
Structure-Guided Modification of Heterocyclic Antagonists of the P2Y14 Receptor | Journal of Medicinal Chemistry
Synthetic RNA Modulators in Drug Discovery | Journal of Medicinal Chemistry
Dehydrozingerone Inspired Styryl Hydrazine Thiazole Hybrids as Promising Class of Antimycobacterial Agents | ACS Medicinal Chemistry Letters
Discovery of Novel BRD4 Ligand Scaffolds by Automated Navigation of the Fragment Chemical Space | Journal of Medicinal Chemistry
Discovery of Imidazole-Based Inhibitors of Plasmodium falciparum cGMP-Dependent Protein Kinase | ACS Medicinal Chemistry Letters
Small Molecules Promote Selective Denaturation and Degradation of Tubulin Heterodimers through a Low-Barrier Hydrogen Bond | Journal of Medicinal Chemistry
Journal of Natural Products Special Issue Honors Drs. Rachel Mata and Barbara N. Timmermann - ACS Axial | ACS Publications
Acute coronary syndromes in diabetic patients, outcome, revascularization, and antithrombotic therapy - ScienceDirect
Synthesis of Thymoquinone–Artemisinin Hybrids: New Potent Antileukemia, Antiviral, and Antimalarial Agents | ACS Medicinal Chemistry Letters
Development of Novel Epoxyketone-Based Proteasome Inhibitors as a Strategy To Overcome Cancer Resistance to Carfilzomib and Bortezomib | Journal of Medicinal Chemistry
Discovery of a 3-(4-Pyrimidinyl) Indazole (MLi-2), an Orally Available and Selective Leucine-Rich Repeat Kinase 2 (LRRK2) Inhibitor that Reduces Brain Kinase Activity | Journal of Medicinal Chemistry
The “Cyclopropyl Fragment” is a Versatile Player that Frequently Appears in Preclinical/Clinical Drug Molecules | Journal of Medicinal Chemistry
